Lorundrostat Shows Promise as New Hypertension Treatment Option

New research presented at the American College of Cardiology Scientific Session 2025 suggests that lorundrostat, an investigational drug, can effectively lower blood pressure in patients with uncontrolled and resistant hypertension.

A phase 2b study, ADVANCE-HTN, evaluated the efficacy and safety of lorundrostat as add-on therapy to standard treatment for patients who remain hypertensive despite taking two to five medications. In total, 285 patients were enrolled in the US trial, who received either a low dose (50mg) or an escalating dose (up to 100mg) of lorundrostat daily.

After 12 weeks, the study found that those receiving the higher dose had a placebo-adjusted reduction in 24-hour average ambulatory blood pressure of 6.5mmHg, while those on the lower dose had a reduction of 7.9mmHg. Lorundrostat was well-tolerated, with side effects consistent with other similar drugs.

The study’s lead author, Dr. Luke Laffin, noted that lorundrostat has a favorable safety profile and may be beneficial for patients with resistant hypertension. Gina Lundberg, another study author, praised the trial’s diversity, which included 40% women and 53% Black participants, as an important aspect of the research.

The addition of lorundrostat to treatment regimens could provide a valuable new option for managing resistant hypertension, although further monitoring is required due to potential side effects.

Source: https://www.medscape.com/viewarticle/advance-htn-shows-benefit-lorundrostat-resistant-2025a10007km?form=fpf